15
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1278 | Astemizole | Laridal,Histaminos,Paralergin | Potassium Channel , Histamine Receptor |
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re... | |||
T4526 | Piperoxan hydrochloride | dl-Piperoxan hydrochloride,Benodaine hydrochloride | Adrenergic Receptor |
Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered. | |||
T6562 | Latrepirdine dihydrochloride | Dimebolin dihydrochloride,Latrepirdine,Latrepirdine 2HCl,Dimebolin | Beta Amyloid , 5-HT Receptor , Adrenergic Receptor , GluR , Autophagy , Histamine Receptor |
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihistamine drug. | |||
T21419 | Diphenhydramine | Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255 | Histamine Receptor |
Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the treatment of allergies. Diphenhydramine is also used in th... | |||
T4563 | Thonzylamine | neohetramine | Histamine Receptor |
Thonzylamine (neohetramine) is an antihistamine and anticholinergic drug. It is available as combination products with Clofedanol or Phenylephrine for temporary relief of symptoms of common cold, hay fever (allergic rhin... | |||
T21390 | Fexofenadine | Carboxyterfenadine,Telfast,MDL 16.455,Allegra | Histamine Receptor |
Fexofenadine (Carboxyterfenadine), an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. Compared to first-generation antihistamines, Fexofenadine is... | |||
T24575 | Oxetorone fumarate | L-6257,L6257,L 6257,Nocertone | |
Oxetorone fumarate is a serotonin antagonist, antihistamine, and alpha-blocker. It was used as an antimigraine drug. | |||
T24851 | Talastine HCl | HL-2186,Talastine hydrochloride,HL2186,Ahanon,HL 2186 | |
Talastine is an antihistamine drug. | |||
T25413 | Fenethazine | RP 3015,Lisergan,Phenetazine,RP-3015,Ethysene | |
Fenethazine is an effective antihistamine used as an antiallergic drug. | |||
T69516 | Thenalidine tartrate | ||
Thenalidine is an antihistamine with anticholinergic properties used as an antipruritic drug. It was withdrawn from the US, Canadian, and UK markets due to a risk of neutropenia. Thenalidine is an antagonist of the H1-re... | |||
T33978 | Phenindamine Tartrate | Pernovine,Thephorin,Nolahist,Phenindamine,Plegine | |
Phenindamine Tartrate is an antihistamine and anticholinergic drug closely related to cyproheptadine. It is used to treat symptoms of the common cold and allergies, such as sneezing, itching, rashes, and hives. | |||
T71537 | Tofenacin hydrochloride | ||
Tofenacin hydrochloride is an antidepressant drug with a tricyclic-like structure. It acts as a serotonin-norepinephrine reuptake inhibitor, and based on its close relation to orphenadrine, may also possess anticholinerg... | |||
T69012 | Cinnarizine clofibrate | ||
Cinnarizine clofibrate is a calcium channel protein inhibitor as well as an antihistamine channel blocker. The compound is a drug derivative of piperazine. Cinnarizine is used for the control of vomiting due to motion si... | |||
T70487 | Tofenacin (free base) | ||
Tofenacin (free base) is an antidepressant drug with a tricyclic-like structure. It acts as a serotonin-norepinephrine reuptake inhibitor, and based on its close relation to orphenadrine, may also possess anticholinergic... | |||
T70247 | Clemizole sulfate | ||
Clemizole sulfate is a drug in clinical development for the treatment of hepatitis C virus (HCV) infection. Clemizole is a novel inhibitor of TRPC5 channels. Clemizole is an H1 antagonist. Clemizole, an antihistamine dru... |